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Atomistry » Silicon » PDB 1fuq-7zpw » 4mpw » |
Silicon in PDB 4mpw: Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone)Enzymatic activity of Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone)
All present enzymatic activity of Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone):
3.4.21.59; Protein crystallography data
The structure of Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone), PDB code: 4mpw
was solved by
A.White,
A.J.Stein,
R.Suto,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Other elements in 4mpw:
The structure of Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone) also contains other interesting chemical elements:
Silicon Binding Sites:
The binding sites of Silicon atom in the Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone)
(pdb code 4mpw). This binding sites where shown within
5.0 Angstroms radius around Silicon atom.
In total 2 binding sites of Silicon where determined in the Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone), PDB code: 4mpw: Jump to Silicon binding site number: 1; 2; Silicon binding site 1 out of 2 in 4mpwGo back to Silicon Binding Sites List in 4mpw
Silicon binding site 1 out
of 2 in the Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone)
Mono view Stereo pair view
Silicon binding site 2 out of 2 in 4mpwGo back to Silicon Binding Sites List in 4mpw
Silicon binding site 2 out
of 2 in the Human Beta-Tryptase Co-Crystal Structure with [(1,1,3,3- Tetramethyldisiloxane-1,3-Diyl)Di-1-Benzofuran-3,5-Diyl]Bis({4-[3- (Aminomethyl)Phenyl]Piperidin-1-Yl}Methanone)
Mono view Stereo pair view
Reference:
S.F.Giardina,
M.Pingle,
K.W.Foreman,
D.S.Werner,
D.E.Bergstrom,
F.Barany,
L.D.Arnold.
Target-Directed Self-Assembly of Homodimeric Drugs To Be Published.
Page generated: Wed Dec 16 02:09:33 2020
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